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Soares, Pedro, Gadd, Morgan S, Frost, Julianty ORCID: 0000-0001-8209-2575, Galdeano, Carles, Ellis, Lucy, Epemolu, Ola, Rocha, Sonia, Read, Kevin D and Ciulli, Alessio (2018) Group-Based Optimization of Potent and Cell-Active Inhibitors of the von Hippel-Lindau (VHL) E3 Ubiquitin Ligase: Structure-Activity Relationships Leading to the Chemical Probe (2<i>S</i>,4<i>R</i>)-1-((<i>S</i>)-2-(1-Cyanocyclopropanecarboxamido)-3,3-dimethylbutanoyI)-4-hydroxy-<i>N</i>-(4-(4-methylthiazol-5-yl)benzyppyrrolidine-2-carboxamide (VH298). JOURNAL OF MEDICINAL CHEMISTRY, 61 (2). pp. 599-618.

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Frost, Julianty ORCID: 0000-0001-8209-2575, Galdeano, Carles, Soares, Pedro, Gadd, Morgan S, Grzes, Katarzyna M, Ellis, Lucy, Epemolu, Ola, Shimamura, Satoko, Bantscheff, Marcus, Grandi, Paola et al (show 4 more authors) , Read, Kevin D, Cantrell, Doreen A, Rocha, Sonia and Ciulli, Alessio (2016) Potent and selective chemical probe of hypoxic signalling downstream of HIF-α hydroxylation via VHL inhibition. Nature communications, 7 (1).

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De Rycker, Manu, Horn, David, Aldridge, Bree, Amewu, Richard K ORCID: 0000-0002-4676-436X, Barry, Clifton EIII, Buckner, Frederick S, Cook, Sarah, Ferguson, Michael AJ, Gobeau, Nathalie, Herrmann, Jennifer et al (show 27 more authors) , Herding, Paul, Hope, William ORCID: 0000-0001-6187-878X, Keiser, Jennifer, Lafuente-Monasterio, Maria Jose, Leeson, Paul D, Leroy, Didier, Manjunatha, Ujjini H, McCarthy, James, Miles, Timothy J, Mizrahi, Valerie, Moshynets, Olena, Niles, Jacquin, Overington, John P, Pottage, John, Rao, Srinivasa PS, Read, Kevin D, Ribeiro, Isabela, Silver, Lynn L, Southern, Jen, Spangenberg, Thomas, Sundar, Shyam, Taylor, Caitlin, Van Voorhis, Wes, White, Nicholas J, Wyllie, Susan, Wyatt, Paul G and Gilbert, Ian H (2020) Setting Our Sights on Infectious Diseases. ACS INFECTIOUS DISEASES, 6 (1). pp. 3-13.

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Zhang, Shaowei, Sakuma, Michiyo, Deora, Girdhar S, Levy, Colin W, Klausing, Alex, Breda, Carlo, Read, Kevin D, Edlin, Chris D, Ross, Benjamin P, Muelas, Marina Wright et al (show 8 more authors) , Day, Philip J, O'Hagan, Stephen, Kell, Douglas B ORCID: 0000-0001-5838-7963, Schwarcz, Robert, Leys, David, Heyes, Derren J, Giorgini, Flaviano and Scrutton, Nigel S (2019) A brain-permeable inhibitor of the neurodegenerative disease target kynurenine 3-monooxygenase prevents accumulation of neurotoxic metabolites. COMMUNICATIONS BIOLOGY, 2 (1). 271-.